Synthesis of two novel mixed bifunctional chelating agents: DO2AP(t Bu) 4and DO3AP(t Bu)4

Fabio Travagin; Luca Biondi; Luciano Lattuada; Giovanni B. Giovenzana

doi:10.1055/s-0040-1707893

Synthesis of two novel mixed bifunctional chelating agents: DO2AP(t Bu) ₄and DO3AP(t Bu)₄

Fabio Travagin
, Luca Biondi
, Luciano Lattuada
, Giovanni B. Giovenzana

Department of Pharmaceutical Sciences

Research output: Contribution to journal › Article › peer-review

Abstract

A convenient synthesis of two novel macrocyclic bifunctional chelating agents (BFCAs), formally derived from the well-known ligands DO3A and DOTA by selective replacement of one carboxymethyl side arm with a phosphonomethyl residue, is reported.

Original language	English
Pages (from-to)	1291-1294
Number of pages	4
Journal	Synlett
Volume	31
Issue number	13
DOIs	https://doi.org/10.1055/s-0040-1707893
Publication status	Published - 28 Jul 2020

Keywords

DO3A
DOTA
bifunctional chelating agents
phosphonic group
protecting group

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10.1055/s-0040-1707893

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title = "Synthesis of two novel mixed bifunctional chelating agents: DO2AP(t Bu) 4and DO3AP(t Bu)4",

abstract = "A convenient synthesis of two novel macrocyclic bifunctional chelating agents (BFCAs), formally derived from the well-known ligands DO3A and DOTA by selective replacement of one carboxymethyl side arm with a phosphonomethyl residue, is reported.",

keywords = "DO3A, DOTA, bifunctional chelating agents, phosphonic group, protecting group",

author = "Fabio Travagin and Luca Biondi and Luciano Lattuada and Giovenzana, \{Giovanni B.\}",

year = "2020",

month = jul,

day = "28",

doi = "10.1055/s-0040-1707893",

language = "English",

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journal = "Synlett",

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T2 - DO2AP(t Bu) 4and DO3AP(t Bu)4

AU - Travagin, Fabio

AU - Biondi, Luca

AU - Lattuada, Luciano

AU - Giovenzana, Giovanni B.

PY - 2020/7/28

Y1 - 2020/7/28

N2 - A convenient synthesis of two novel macrocyclic bifunctional chelating agents (BFCAs), formally derived from the well-known ligands DO3A and DOTA by selective replacement of one carboxymethyl side arm with a phosphonomethyl residue, is reported.

AB - A convenient synthesis of two novel macrocyclic bifunctional chelating agents (BFCAs), formally derived from the well-known ligands DO3A and DOTA by selective replacement of one carboxymethyl side arm with a phosphonomethyl residue, is reported.

KW - DO3A

KW - DOTA

KW - bifunctional chelating agents

KW - phosphonic group

KW - protecting group

UR - https://www.scopus.com/pages/publications/85089500454

U2 - 10.1055/s-0040-1707893

DO - 10.1055/s-0040-1707893

M3 - Article

SN - 0936-5214

VL - 31

SP - 1291

EP - 1294

JO - Synlett

JF - Synlett

IS - 13

ER -

Synthesis of two novel mixed bifunctional chelating agents: DO2AP(t Bu) ₄and DO3AP(t Bu)₄

Abstract

Keywords

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